Robert R. Fenichel |
Therapeutic Level (µM) | ||||
---|---|---|---|---|
Drug | Total | Free | Ref | Comment |
amiodarone | 1-4 | 0.001 | 8 | |
amitriptyline | 0.2-0.7 | 0.02 | 9 | |
astemizole | 0.002-0.003 | 25 | ||
desmethylastemizole | 0.02 | 25 | ||
buprenorphine | 0.036 | 71 | secondary reference | |
captopril | 0.23 | 0.15 | 10 | |
cetirizine | 0.67 | 0.07 | 1 | |
chlorpromazine | 0.1-1.1 | 17 | controversial | |
cisapride | 0.05-0.2 | 48 | ||
clarithromycin | 2.7-4 | 1.5-2 | 67 | |
codeine | 0.66 | 71 | secondary reference | |
diphenhydramine | 0.09 | 0.02 | 11 | |
disopyramide | 15 | 130 | ||
EDDP | 1 | 71 | secondary reference | |
erythromycin | 13.6 | 67 | intravenous | |
fentanyl | 0.03 | 71 | secondary reference | |
LAAM | 1 | 71 | secondary reference | |
meperidine | 1.3 | 71 | secondary reference | |
methadone | 3.6 | 71 | secondary reference | |
morphine | 2.5 | 71 | secondary reference | |
ranolazine | 5.8 | 6 |